发明名称 Heterocyclic compounds.
摘要 <p>A compound of the formula (I) &lt;CHEM&gt; or an acid addition salt thereof, wherein R is hydrogen or C1-4 alkyl, R&lt;1&gt; is chlorine or methyl optionally substituted by one or two fluorine, R&lt;2a&gt; to R&lt;2d&gt; are the same or different and are chosen from the group comprising hydrogen, chlorine, bromine, fluorine, C1-4 alkyl optionally substituted by fluorine or chlorine atoms, C1-4 alkoxy, C1-4 acyl, C1-4 alkoxycarbonyl, C1-4alkylthio, nitro, cyano, amino optionally substituted by C1-4 alkyl or C1-4 acyl; E is C6-10 aryl or aralkyl, a group CH2C (Me)2OR&lt;3&gt; wherein R&lt;3&gt; is hydrogen, C1-4 acyl, C1-4 alkyl or C2-8 carbamyl, a group CH=C(Me)CH2CH2CH=CMe2, a group - @@ @@Me2, a group OCHR&lt;4&gt;R&lt;5&gt; wherein R&lt;4&gt;and R&lt;5&gt; are the same or different and each is methyl or ethyl, a group CH=CR&lt;6&gt;R&lt;7&gt; wherein R&lt;6&gt; is hydrogen, chlorine, bromine, fluorine, C1-4 alkyl, C1-8 alkoxycarbonyl, C1-4 alkynyl or C1-8 acyl and R&lt;7&gt; is hydrogen, chlorine, bromine, fluorine or C1-4 alkyl, or a group CH=X-Y-R&lt;8&gt; wherein X is N or C(R&lt;9&gt;) wherein R&lt;9&gt; is hydrogen or C1-6alkyl, Y is oxygen, sulphur or a group NR&lt;1&gt;&lt;0&gt; wherein R&lt;1&gt;&lt;0&gt; is C1-8 hydrocarbyl, R&lt;8&gt; is C1-4 acyl or C1-10 hydrocarbyl optionally substituted by C1-4 alkyl, C1-4 alkoxy, C1-4 acyl or halogen, or, when X is nitrogen, R&lt;8&gt; may be hydrogen; provided that at least of of R&lt;2a&gt; to R&lt;2d&gt; is other than hydrogen when R&lt;1&gt; is methyl or chlorine except when E is OCHR&lt;4&gt;R&lt;5&gt;, C6-10 aryl and aralkyl, CH=CR&lt;6&gt;R&lt;7&gt; or CH=XYR&lt;8&gt; or R&lt;3&gt; is C2-8 carbamyl and that R&lt;2c&gt; is not methyl when R&lt;1&gt; is methyl except when E is CH=CR&lt;6&gt;R&lt;7&gt; or CH=XYR&lt;8&gt;, and other than 1-geranyl-2-methylbenzimidazole, processes for their preparation, formulations containing them and their use in the control of pests, helminths and fungi.</p>
申请公布号 EP0269230(A1) 申请公布日期 1988.06.01
申请号 EP19870308918 申请日期 1987.10.08
申请人 THE WELLCOME FOUNDATION LIMITED 发明人 WESTON, JOHN BERNARD;PULMAN, DAVID ALLEN;FRENKEL, ALEXANDER DAVID
分类号 C07D235/08;C07D235/24;C07D405/06 主分类号 C07D235/08
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