发明名称 Förfarande för framställning av nya terapeutiskt användbara 7-/2-(2-am inotiazol-4-yl)iminoacetamido/cefalosporinderivat.
摘要 <p>Compounds of the formula <IMAGE> I wherein R1 is hydrogen or a conventional amino-protecting group, R2 and R3 each are independently methyl or ethyl, and R4 is methyl, ethyl, n-propyl, isopropyl, n-butyl, isobutyl, allyl, 2-butenyl, 3-butenyl, 2-hydoxyethyl, 3-hydroxypropyl, 2-(dimethylamino)ethyl, pyridylmethyl, pyridylethyl, benzyl or phenethyl, and nontoxic pharmaceutically acceptable acid addition salts and solvates thereof, as well as processes for their preparation, are disclosed. The compounds in which R1 is hydrogen are potent antibacterial agents.</p>
申请公布号 FI74974(C) 申请公布日期 1988.04.11
申请号 FI19830001013 申请日期 1983.03.24
申请人 BRISTOL-MYERS CO, 发明人 KAMACHI,HAJIME;OKUMURA,JUN;NAITO,TAKAYUKI
分类号 C07D501/06;A61K;A61K31/34;A61K31/45;A61K31/545;A61K31/546;A61P31/04;C07D;C07D501/00;C07D501/02;C07D501/16;C07D501/20;C07D501/24;C07D501/38;C07D501/46;(IPC1-7):C07D501/46 主分类号 C07D501/06
代理机构 代理人
主权项
地址
您可能感兴趣的专利