发明名称 |
DERIVATIVES OF CERVINOMYCIN ANTIBIOTICS AND PROCESS FOR THEIR PREPARATION. |
摘要 |
<p>Cervinomycin derivs. of formula (I) are new: where at least one of R1, R2 and R3 is acyl or alkyl and the rest are H; R4 is H or alkyl; B is a ring moiety of formula (II) or (III). Reaction of cervinomycin A2 (I, R1 = R4 = H, B is (II)) or cervinomycin A1 (I, R1 = R2 = R3 = R4 = H, B is (III)) with an alkylating or acylating agent.</p> |
申请公布号 |
EP0259496(A1) |
申请公布日期 |
1988.03.16 |
申请号 |
EP19870901638 |
申请日期 |
1987.02.17 |
申请人 |
THE KITASATO INSTITUTE |
发明人 |
OMURA, SATOSHI 12-7, SETA 5-CHOME;NAKAGAWA, AKIRA SUMIYOSHI JUTAKU 4-206;IWAI, YUZURU 9-303, 2-1 KARABE 2-CHOME |
分类号 |
C07D498/04;A61K31/435;A61P31/04;C07D498/14 |
主分类号 |
C07D498/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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