发明名称 DERIVATIVE OF PYRAZOLE, INSECTICIDE COMPRISING THEREOF AS ACTIVE COMPONENT, INTERMEDIATE COMPOUND, METHODS FOR PREPARING COMPOUNDS
摘要 FIELD: organic chemistry, insecticides, chemical technology. ^ SUBSTANCE: invention describes derivative of 1-aryl-3-cyano-5-heteroarylalkylaminopyrazole of the general formula (1): wherein A means: (A-1) , (A-2) , (A-3) and (A-4) and wherein X represents C-halogen; R1 represents (C1-C4)-alkyl group or halogen-(C1-C4)-alkyl group; A represents any group among (A-1) - (A-4) wherein R4 represents hydrogen atom or (C1-C4)-alkyl group; n = 0, 1 or 2 under condition that R1 represents halogen-(C1-C4)-alkyl group with exception for perhalogenalkyl group when A represents (A-1) and n = 0, and that n doesn't equal 0 when A represents (A-4). Also, invention describes derivative of pyrazole of the formula (2): wherein A means: (A-1) and Y means: (Y-1) , (Y-2) and (Y-3) wherein X, R2, R3 and R4 have values given above; R5 represents hydrogen atom; A represents (A-1); Y means any group among (Y-1) - (Y-3); Z represents halogen atom that are intermediate compounds used for synthesis of the compound (1). Invention describes methods for preparing compounds of the formula (1) and (2) and insecticide comprising compound of the formula (1) as an active component. Insecticide shows high systemic activity, high safety and reduced harmful effect on environment in vicinity areas of its applying. ^ EFFECT: improved methods for preparing, valuable insecticide properties of compound. ^ 11 cl, 9 tbl, 19 ex
申请公布号 RU2256658(C2) 申请公布日期 2005.07.20
申请号 RU20010135851 申请日期 2000.06.28
申请人 发明人 OKUI SUKO;KIOMURA NOBUO;FUKUTI TOSIKI;TANAKA KEN;KATSURADA MANABU;OKANO KAZUJA;SUMITANI NAOKO;MIJAUTI AKIKO;JABE AKIKO
分类号 A01N43/56;A01N43/58;A01N43/60;A01N47/02;C07D401/12;C07D403/12 主分类号 A01N43/56
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