发明名称 VERFAHREN ZUR HERSTELLUNG VON THIAZOLE(4,5-C)CHINOLIN-DERIVATEN
摘要 The invention relates to new thiazolo[4,5-c]quinoline derivatives of the general Formula I <IMAGE> (I) and acid addition salts thereof, a process for the preparation of the same and pharmaceutical compositions comprising the said compounds. The substituent definition of the general Formula I is as follows: R stands for hydrogen; a straight or branched chained alkyl group having 2-5 carbon atoms optionally substituted by one or more halogen atom(s); phenyl or phenyl-(lower alkyl) optionally bearing one or more substituent(s) on the phenyl ring; R1 and R2 are identical or different and stand for hydrogen, halogen or lower alkyl). The compounds of the general Formula I possess valuable central nervous depressive properties.
申请公布号 DD254202(A5) 申请公布日期 1988.02.17
申请号 DD19860296208 申请日期 1986.11.12
申请人 EGIS GYOGYSZERGYAR 发明人 KNOLL,JOZSEF;BERENYI,EDIT;BUDAI,KATALIN;KNOLL,BERTA;FUERTS,ZSUZSA;TIMBR,JULIA;ZSILA,GABRIELLA;NIKLYA,ILDIKO;PETOCZ,LUJZA;MANDI,ATTILA
分类号 A61K31/47;A61K31/4738;A61P25/22;A61P25/24;A61P25/26;C07D513/04;(IPC1-7):C07D513/04;C07D215/02;C07D277/00 主分类号 A61K31/47
代理机构 代理人
主权项
地址