Method for preparing substituted triazolopyridines

摘要

The present invention relates to methods of preparing substituted triazolopyridine compounds of general formula (I) as described and defined herein, as well as to intermediate compounds useful in the preparation of said compounds.;

主权项

1. Method for preparing a compound of formula (I): comprising reacting a compound of formula (In1): with a compound of formula (In5) wherein one of the groups CG1 and CG2 represents chloro, bromo, iodo or trifluoromethylsulfonyloxy, and the other one of the groups CG1 and CG2 represents a boronic acid or an ester thereof, thus providing the compound of formula (I).