发明名称 SPIROKVATERNAERA AMMONIUMHALOGENIDER OCH N-(2-PYRIMIDINYL)PIPERAZINYLALKYLAZASPIROALKANDIONPROCESS.
摘要 Novel spiro-quaternary ammonium halides are disclosed. The new compounds are particularly valuable as intermediates in preparation of N-(2-pyrimidinyl)piperazinylalkyl derivatives of azaspiroalkanediones such as the psychopharmacologic agent 8-[4-[4-(2-pyrimidinyl)-1-piperazinyl]butyl]-8-azaspiro[4.5]decane-7,9 -dione.
申请公布号 FI75159(B) 申请公布日期 1988.01.29
申请号 FI19810003178 申请日期 1981.10.13
申请人 BRISTOL-MYERS COMPANY 发明人 SIMMS, JACK C.
分类号 C07D401/12;C07D471/10;C07D487/10 主分类号 C07D401/12
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