发明名称 Isoxazolone derivatives and production thereof.
摘要 <p>The present invention related to a compound of the formula : &lt;CHEM&gt; wherein R&lt;1&gt; is hydrogen, isonitrile or an organic residue bonded through nitrogen ; R is hydrogen, alkyl which may be substituted, alkylthio in which sulfur atom may be oxidized or azido, or forms a double bond together with the adjacent carbon atom; provided that when R&lt;1&gt; is an organic residue bonded through nitrogen, R is not hydrogen; R&lt;2&gt; is carboxyl or a group derivable therefrom, and a salt thereof, and a method for producing the same. The Compound (I) of the present invention has, among others, an excellent anitimicrobial activity and is useful as an antimicrobial agent, etc.</p>
申请公布号 EP0250096(A1) 申请公布日期 1987.12.23
申请号 EP19870304458 申请日期 1987.05.20
申请人 TAKEDA CHEMICAL INDUSTRIES, LTD. 发明人 MASUYA, HIROTOMO
分类号 A61K38/00;C07D413/04;A61K31/42;A61K31/425;A61P31/04;C07D417/14;C07K5/078 主分类号 A61K38/00
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