发明名称 SUBSTITUTED DIHYDROIMIDAZO(1,2-A)QUINOXALINES
摘要 This invention relates to a novel class of substituted dihydroimidazo [1,2-a] quinoxaline derivatives of the formula …<CHEM>… wherein… R<1> is C1-C6 alkyl, benzyl, phenyl, a …<CHEM>… group, a ……(NH2-@-CH2)-… group or a ……(R<5>-@)-… group wherein R<4> is C1-C6 alkyl, and R<5> is C1-C8 alkyl, aminomethyl, pyridinyl, phenyl, halophenyl or a ……(R<6>-O-@-NHCH2)- group wherein R<6> is C1-C6 alkyl;… R<2> is phenyl or substituted phenyl having 1 or 2 substituents selected from the class consisting of halo or C1-C6 alkoxy;… R<3> is hydrogen or halogen; and… X is -CH- or -N-… and to pharmaceutical compositions containing such compounds. The compounds and compositions are effective as anti-anaerobic agents.
申请公布号 ZA8606805(B) 申请公布日期 1987.11.25
申请号 ZA19860006805 申请日期 1986.09.08
申请人 G.D. SEARLE & CO. 发明人 GEORGE JOHN ELLAMES;ALBERT ANDREJ JAXA-CHAMIEC
分类号 A61K31/495;A61P31/04;C07D471/14;C07D487/04 主分类号 A61K31/495
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