发明名称 |
ANTI-IMFLAMMATORY POLYMORPHIC MONOETHANOLAMINE SALT OF N-(2-PYRIDYL)-2-METHYL-4-HYDROXY-2H-1,2-BENZOTHIAZINE-3-CARBOXAMIDE 1,1-DIOXIDE COMPOUND; COMPOSITION AND METHOD OF USE THEREFOR |
摘要 |
A novel crystalline form of the monoethanolamine salt of N-(2-pyridyl)-2-methyl-4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide has been prepared. This novel crystalline form is designated as polymorph I and is useful in therapy as a non-steroidal anti-arthritic agent. Methods for preparing this polymorph from readily available materials are provided. |
申请公布号 |
PH21322(A) |
申请公布日期 |
1987.09.28 |
申请号 |
PH19580000330 |
申请日期 |
1985.11.15 |
申请人 |
PFIZER INC. |
发明人 |
ROBERTSON ROBERT LEE |
分类号 |
C07D279/16;A61K31/44;A61K31/54;A61K31/5415;A61P29/00;C07D417/12;F16L57/00 |
主分类号 |
C07D279/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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