发明名称 |
Prodrug compounds, process for the preparation thereof and sustained release preparation comprising the same. |
摘要 |
<p>A Prodrug compound of the formula :
A-CO(CH2)m(NHCO)n-R
wherein A is a residue of pharmaceutical compound having @@NH or -NH2 group in the molecule,
R is a residue of steroid compound,
m is an integer of l to 5 and
n is 0 or l,
and its salts, process for its preparation and a sustained release preparation comprising it. </p> |
申请公布号 |
EP0237051(A2) |
申请公布日期 |
1987.09.16 |
申请号 |
EP19870103518 |
申请日期 |
1987.03.11 |
申请人 |
FUJISAWA PHARMACEUTICAL CO., LTD. |
发明人 |
HASHIMOTO, MASASHI;TAKENO, HIDEKAZU;KAYAKIRI, HIROSHI;KAGAYAMA, AKIRA;TOKUNAGA, YUJI;IWASA, TOMOAKI |
分类号 |
C07H21/00;C07J43/00;(IPC1-7):C07J43/00;A61K31/58 |
主分类号 |
C07H21/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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