发明名称 PROCEDIMIENTO PARA PREPARAR 5H,11H-PIRROLO (2,1-C)(1,4)BENZOXAZEPINAS SUSTITUIDAS EN POSICION 11
摘要 <p>There are described to novel 11-substituted 5H,11H-pyrrolo[2,1-c] [1,4]benzoxazepines of the general formula <CHEM> where m and n are each independently, 0, 1 or 2 and m + n is 1 or 2, X and Y are each independently hydrogen, loweralkyl or halogen, and R is hydrogen, cyano, <CHEM> unsubstituted loweralkyl, or substituted loweralkyl having one to three substituents each of which being independently cyano, hydroxy, cyclohexyl, furyl, <CHEM> k being 1, 2 or 3, W being each independently hydrogen, halogen, hydroxy, loweralkyl, trifluoromethyl, loweralkoxy, nitro, amino, diloweralkylamino, phenoxy, or benzyloxy, and Z being hydrogen, loweralkyl or halogen, which are useful as antipsychotic and analgesic agents; novel intermediate compounds therefor; and methods of synthesizing the foregoing compounds.</p>
申请公布号 ES552578(D0) 申请公布日期 1987.09.16
申请号 ES19780005525 申请日期 1986.03.01
申请人 HOECHST-ROUSSEL PHARMACEUTICAL INCORPORATED 发明人
分类号 A61K31/00;A61K31/55;A61P25/04;A61P25/18;A61P25/24;A61P25/26;C07D207/32;C07D207/333;C07D401/06;C07D498/04;(IPC1-7):C07D413/04 主分类号 A61K31/00
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