发明名称 STEROID DERIVATIVE AND PRODUCTION THEREOF
摘要 NEW MATERIAL:A compound expressed by formula I [formula II represents formula III or IV; R1 represents lower alkyl; R2 represents lower alkyl, lower alkoxyalkyl, tetrahydropyranyl or formula V (R4-R6 represent lower alkyl or phenyl); R3 represents lower alkyl]. EXAMPLE:A compound expressed by formula VI. USE:A raw material for pavoninin of shark-repelling substance. PREPARATION:A compound expressed by formula VII is hydrogenated to produce a compound expressed by formula VIII, which is reacted with a compound expressed by the formula R3-CH2COY1 (Y1 represents halogen atom). Then the obtained compound is reacted with a strong base, then with a compound expressed by formula IX (Y2 represents halogen atom) and further subjected to Claisen rearrangement reaction to obtain a compound expressed by formula X, and the formula XI of this compound is reduced, and this compound is hydrolized.
申请公布号 JPS62205100(A) 申请公布日期 1987.09.09
申请号 JP19860044262 申请日期 1986.03.03
申请人 NIPPON KAYAKU CO LTD 发明人 NAKAI TAKESHI;MIKAMI KOICHI
分类号 C07J9/00 主分类号 C07J9/00
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