摘要 |
Phenylbutene derivatives having optionally substituted phenyl and pyrrolyl, furanyl, pyridinyl, pyrazinyl, imidazolyl, pyrazolyl, pyrimidinyl, pyrrolodinyl, tetrahydrofuranyl, piperidinyl, piperazinyl or alkylthienyl in the 4-position and 3-carboxypiperid-1-yl, 3-carboxytetrahydropyrid-1-yl or 3-carboxymethylpyrrolidin-1-yl in the 1-position potentiate GABA min ergic neurotransmission. |