发明名称 |
PROCESS FOR PREPARING CHIRAL BETA-ADRENOCEPTOR ANTAGONISTS AND INTERMEDIATES THEREOF |
摘要 |
The S-isomer of a compound of the formula (V), wherein Ar is an optionally substituted aryl, heteroaryl or heterocyclic group, and R<1> is phenyl optionally substituted by C1-6alkoxy or C1-6alkyl and its use in a process for the preparation of the S-isomer of compounds of formula (VII), wherein the group R<2>R<3>CH- is optionally substituted alkyl. |
申请公布号 |
ZA8508363(B) |
申请公布日期 |
1987.06.24 |
申请号 |
ZA19850008363 |
申请日期 |
1985.10.31 |
申请人 |
SMITH KLINE & FRENCH LABORATORIES LIMITED |
发明人 |
JOHN KITTERINGHAM;MICHAEL BARRY MITCHELL |
分类号 |
C07C217/32;A61K31/045;A61K31/085;A61K31/13;A61K31/135;A61K31/33;A61K31/40;A61K31/41;A61K31/47;C07C;C07C43/00;C07C67/00;C07C213/00;C07D209/00;C07D209/43;C07D213/00;C07D213/63;C07D215/20;C07D239/34;C07D263/00;C07D263/04;C07D263/06;C07D263/20;C07D263/24;C07D285/10;C07D295/08 |
主分类号 |
C07C217/32 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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