发明名称 |
Azetidinone derivative and process for preparing the same. |
摘要 |
<p>An azetidinone derivative having the general formula (I):
<Chemistry id="chema01" num="0001"><Image id="ia01" he="44" wi="110" file="IMGA0001.TIF" imgContent="chem" imgFormat="TIFF" /></Chemistry> wherein R¹ and R² are hydrogen atom or a protective group and R³ is an alkyl group or hydrogen atom, a process for preparing the same, and a process for preparing an azetidinone derivative having the general formula (II):
<Chemistry id="chema02" num="0002"><Image id="ia02" he="42" wi="125" file="IMGA0002.TIF" imgContent="chem" imgFormat="TIFF" /></Chemistry> wherein R¹, R² and R³ are as above. The azetidinone derivative (I) of the present invention can be converted into an important intermediate of lβ-methylcarbapenem antibiotics by a selective reduction of the double bond. </p> |
申请公布号 |
EP0224059(A1) |
申请公布日期 |
1987.06.03 |
申请号 |
EP19860114952 |
申请日期 |
1986.10.28 |
申请人 |
SAGAMI CHEMICAL RESEARCH CENTER |
发明人 |
SHIBASAKI, MASAKATSU;IIMORI, TAKAMASA |
分类号 |
B01J23/00;B01J23/40;C07B61/00;C07D205/08;C07F7/18;(IPC1-7):C07D205/08;C07B53/00 |
主分类号 |
B01J23/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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