发明名称 |
Novel cyclic Hexapeptide LHRH antagonists |
摘要 |
Novel peptides of the formula: <IMAGE> I where R1 through R8 are various radicals derived from L- and D- amino acids; having LHRH antagonist activity; useful in reducing fertility. Pharmaceutical compositions and methods for use in reducing fertility.
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申请公布号 |
US4659691(A) |
申请公布日期 |
1987.04.21 |
申请号 |
US19850699778 |
申请日期 |
1985.02.08 |
申请人 |
MERCK & CO., INC. |
发明人 |
VEBER, DANIEL F.;FREIDINGER, ROGER M. |
分类号 |
C07K7/64;A61K38/00;A61K38/04;A61K38/22;A61P5/00;C07K7/23;C07K14/575;(IPC1-7):A61K37/43;C07K5/12;C07K7/20 |
主分类号 |
C07K7/64 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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