发明名称 Novel cyclic Hexapeptide LHRH antagonists
摘要 Novel peptides of the formula: <IMAGE> I where R1 through R8 are various radicals derived from L- and D- amino acids; having LHRH antagonist activity; useful in reducing fertility. Pharmaceutical compositions and methods for use in reducing fertility.
申请公布号 US4659691(A) 申请公布日期 1987.04.21
申请号 US19850699778 申请日期 1985.02.08
申请人 MERCK & CO., INC. 发明人 VEBER, DANIEL F.;FREIDINGER, ROGER M.
分类号 C07K7/64;A61K38/00;A61K38/04;A61K38/22;A61P5/00;C07K7/23;C07K14/575;(IPC1-7):A61K37/43;C07K5/12;C07K7/20 主分类号 C07K7/64
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