发明名称 PROCESS FOR PREPARING TRIAZOL DERIVATIVES
摘要 <p>Triazol derivs. of formula (I) and its pharmaceutically (or agriculturally) acceptable salts are prepd. by reacting a 1,2,4triazol or its base salt with (II) at 50-130 deg C. m is 0,1,2,3, or 4; n is 0,1,2,3, or 4; Q is leaving gp. e.g. Cl, Br, I, CF3SO2O-, p-toluene sulfonyl oxy. (I) are useful as anti-fungus agent. (II) is obtd. from rxn. of CF3(CF2)nMgI or CF3(CF2nMgBr with QCH2CO(CF2)mCF3.</p>
申请公布号 KR870000786(B1) 申请公布日期 1987.04.18
申请号 KR19840000395 申请日期 1984.01.28
申请人 PFIZER CORP. 发明人 RICHARDSON KENNETH;WHITTLE PETER J.
分类号 A01N43/653;A61K31/41;A61P31/04;C07C29/40;C07D249/08;C07D521/00;(IPC1-7):C07D249/08 主分类号 A01N43/653
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