Esters of boron analogues of amino acids

摘要

Ester analogues of boron analogues of amino acid are disclosed. Also disclosed is a method of forming the ester analogues in high yield by condensation of the corresponding acids and alcohols with dicylohexylcarbodiimide at room temperature in dichloromethane. The disclosed compounds have shown interesting biological activities, in particular, hypolipidemic activity as well as significant antitumor and antiarthritic activities.