发明名称 PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE BENZODIA- ZEPINA
摘要 <p>Benzodiazepine derivs. of formula (I) in which R, is H or lower alkyl for use as tranquillisers or intermediates, are made by reaction of 7-chloro 1-methyl 5-phenyl 3H-1, 4-benzodiazepin 2(1H)-one with a cpd. of formula (II), in organic solvent in presence of a reactive bromine acceptor, at ambient temp.</p>
申请公布号 ES550600(D0) 申请公布日期 1987.03.01
申请号 ES20000005506 申请日期 1985.12.31
申请人 ASTUR PHARMA 发明人
分类号 A61K31/55;C07D243/26;(IPC1-7):C07D243/26 主分类号 A61K31/55
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