发明名称 PROCESS FOR THE PRODUCTION OF SEMI SYNTHETIC STATINS VIA NOVEL INTERMEDIATES
摘要 A process has been provided to produce semi synthetic statins, as for instance simvastatin with a high yield, from another statin, preferably a naturally occurring statin, as for instance lovastatin. Also a number of novel intermediate compounds, prepared during said process, has been provided.
申请公布号 WO9832751(A1) 申请公布日期 1998.07.30
申请号 WO1998EP00519 申请日期 1998.01.27
申请人 GIST-BROCADES B.V.;VRIES, TON, RENE;WIJNBERG, HANS;FABER, WIJNAND, SJOURD;KALKMAN-AGAYN, VENETKA, IVANOVA;SIBEYN, MIEKE 发明人 VRIES, TON, RENE;WIJNBERG, HANS;FABER, WIJNAND, SJOURD;KALKMAN-AGAYN, VENETKA, IVANOVA;SIBEYN, MIEKE
分类号 C07D319/06;A61K31/366;A61K31/39;A61K31/6615;A61P3/08;A61P43/00;C07C231/02;C07C235/26;C07D309/30;C07D327/10;C07F5/02;C07F9/6574;(IPC1-7):C07D309/30;C07C235/30;C07F9/657 主分类号 C07D319/06
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