发明名称 NOVEL ANTIBIOTIC DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND USE THEREOF
摘要 Compounds represented by formula (I), (wherein R<1> represents amino or an organic residue bound via nitrogen, R<2> represents carboxy or its derivative, and X represents hydrogen, methoxy or formylamino, provided that, when R<1> represents acetylamino or amino and X represents hydrogen, R<2> does not represent p-nitrobenzyloxycarbonyl nor benzhydryloxycarbonyl) and salts thereof possess an excellent antibacterial effect, thus being used as antibacterial agents.
申请公布号 WO8700178(A1) 申请公布日期 1987.01.15
申请号 WO1985JP00358 申请日期 1985.06.25
申请人 TAKEDA CHEMICAL INDUSTRIES, LTD. 发明人 YOSHIOKA, KOICHI;HARADA, SETSUO;OCHIAI, MICHIHIKO
分类号 A61K31/42;A61K31/44;A61K31/495;A61K31/50;A61K31/505;A61K31/535;A61K31/55;A61K31/675;A61K31/695;A61K38/00;A61P31/04;C07D237/00;C07D247/00;C07D261/00;C07D307/00;C07D333/00;C07D407/00;C07D413/04;C07D413/14;C07D417/14;C07D521/00;C07F7/08;C07F7/10;C07F9/6539;C07F9/6558;C07K5/06;C12P17/16;C12R1/01 主分类号 A61K31/42
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