发明名称 SUBSTITUTED DODECAHYDROTRIPHENYLENES, DECAHYDRO-1H-CYCLOPENTA(1)PHENANTHRENES, DECAHYDRO-1H-PYRIDO(1,2-F)PHENANTHRIDINES AND DECAHYDROPYRROLO(1,2-F)PHENANTHRIDINES AS CNS AGENTS
摘要 1,2,3,4,4a,4b,5,6,7,8,8a,12b-Dodecahydro-7-(oxo, hydroxy or amino)-9-hydroxy-11-(alkyl, alkoxy or alkoxyalkyl)triphenylenes, 2,3,3a,3b,4,5,6,7,7a,11b-decahydro-6-(oxo, hydroxy or amino)-8-hydroxy-10-(alkyl, alkoxy or alkoxyalkyl)-1H-cyclopenta[1]phenanthrenes, 2,3,4,4a,4b,5,6,7,8,8a-decahydro-7-(oxo, hydroxy or amino)-9-hydroxy-11-(alkyl, alkoxy, alkoxyalkyl, aralkyl, aralkoxy, aryloxyalkyl or aralkoxyalkyl)-1H-pyrido[1,2-f]phenanthridines, and 1,2,3,3a,3b,4,5,6,7,7a-decahydro-6-(oxo, hydroxy or amino)-8-hydroxy-10-(alkyl, alkoxy or alkoxyalkyl)pyrrolo[1,2-f]phenanthridines and derivatives are valuable as central nervous system active agents or as intermediates to compounds having such activity.
申请公布号 DE3367917(D1) 申请公布日期 1987.01.15
申请号 DE19833367917 申请日期 1983.03.09
申请人 PFIZER INC. 发明人 EGGLER, JAMES FREDERICK;MELVIN, LAWRENCE SHERMAN;JOHNSON, MICHAEL ROSS
分类号 C07C69/03;A61K31/05;A61K31/085;A61K31/12;A61K31/135;A61K31/16;A61K31/165;A61K31/215;A61K31/22;A61K31/47;A61K31/475;A61P1/08;A61P1/12;A61P7/10;A61P11/14;A61P25/00;A61P25/04;A61P25/18;A61P25/20;A61P27/02;A61P27/06;C07C27/00;C07C29/09;C07C29/10;C07C29/44;C07C29/56;C07C33/20;C07C39/17;C07C39/42;C07C41/00;C07C43/14;C07C43/174;C07C43/178;C07C43/20;C07C43/23;C07C45/00;C07C49/703;C07C49/727;C07C49/753;C07C49/755;C07C59/72;C07C67/00;C07C69/017;C07C69/035;C07C69/157;C07C69/78;C07C205/32;C07C205/33;C07C213/00;C07C217/74;C07C219/26;C07C227/00;C07C229/06;C07C231/00;C07C233/23;C07C311/07;C07D207/08;C07D211/34;C07D215/22;C07D215/233;C07D455/03;C07D455/04;C07D455/06;C07D471/04;(IPC1-7):C07D455/04;C07C131/00;C07C93/26;C07C103/42;C07C103/80 主分类号 C07C69/03
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