发明名称 FOERFARANDE FOER FRAMSTAELLNING AV TERAPEUTISKT ANVAENDBARA PYRIDOBENSOTIAZINDERIVAT.
摘要 Pyridobenzothiazine derivatives with high antimicrobial activity having the following general formula: …<CHEM>… wherein… R is H or CH3; n is 0 or 1 or 2 and Y is Cl or F, …<CHEM>… wherein R<1> is a C1-C6 alkyl… or a C2-C6 alkenyl, or an arylalkyl, arylalkylcarbonyl, alkylcarbonyl, alkyloxycarbonyl, possibly substituted with halogens or hydroxy groups. …<??>The present invention relates also to the processes for obtaining the compounds having the general formula (I). Such processes consist in synthesis routes using as starting products 3-chloro-4-fluoraniline, or 2,3,4-trifluoronitrobenzene.
申请公布号 FI850741(L) 申请公布日期 1985.08.25
申请号 FI19850000741 申请日期 1985.02.22
申请人 MEDIOLANUM FARMACEUTICI SRL 发明人 MASCELLANI, GIUSEPPE;FRAVOLINI, ARNALDO;TERNI, PATRIZIA
分类号 A61K31/54;A61P31/04;C07D277/82;C07D279/16;C07D513/06 主分类号 A61K31/54
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