发明名称 |
Synthesis of cyclopropane amino acids |
摘要 |
Cyclopropane ("Cyclopropyl") amino acids and peptides containing at least one cyclopropyl amino acid are disclosed. The processes for synthesizing cyclopropyl amino acids and peptides containing at least one cyclopropyl amino acid are also disclosed. Cyclopropyl amino acids are useful as enzyme inhibitors and as substitutes for natural amino acids in peptide hormones such as regulators of bodily functions to enhance bioactivity, to stabilize the peptide into which it is incorporated to cleavage by enzymes and to convert such peptides into enzyme inhibitors.
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申请公布号 |
US4629784(A) |
申请公布日期 |
1986.12.16 |
申请号 |
US19840677901 |
申请日期 |
1984.12.05 |
申请人 |
THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. |
发明人 |
STAMMER, CHARLES H. |
分类号 |
A23L1/236;C07D231/44;C07D403/04;C07K5/072;C07K5/083;C07K5/097;(IPC1-7):C07K5/08;C07K5/10;C07K7/06 |
主分类号 |
A23L1/236 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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