发明名称 PROCESS FOR THE PREPARING OF HEXAHYDRO-TRANS-PYRIDOINDOLE DERIVATIVES
摘要 The title compds. (I) were prepd. by the reaction of (II) and D-(CH2) n-G1. In (I) n is 2-6; D is Cl, Br, I, or CH3SO2O-; G1 is (III), (IV) , (V). (I) are neuroleptic agents used in the treatment of mental disorders and illnesses including schizophrenia, psychoses and neuroses. They exhibit major tranquillizing activity but have fewer side effects than currently used drugs. They may be given orally or parenterally. Dose is typically 0.1-100 mg/day.
申请公布号 KR860001819(B1) 申请公布日期 1986.10.24
申请号 KR19820000154 申请日期 1982.01.15
申请人 PFIZER INC. 发明人 WALTZ, WILLARD M.;HUBERT, CHARLES A.
分类号 C07D471/00;A61K31/435;A61K31/445;A61K31/495;A61P25/02;A61P25/18;A61P25/20;C07D249/12;C07D471/04;(IPC1-7):C07D471/04 主分类号 C07D471/00
代理机构 代理人
主权项
地址