发明名称 UN PROCEDIMIENTO PARA PREPARAR UN DERIVADO DE 1,3-BENZOTIA- ZOL-2(3H)-ONA O 1,3-BENZOXAZOL-2(3H)-ONA
摘要 <p>Compounds of formula (I): …<CHEM>… O-C2-6-alkanoyl derivatives thereof and pharmaceutically acceptable salts are described in which X is -S- or -O-, R<1> and R<2> are, each, hydrogen, C1-6-alkyl, allyl, benzyl, phenethyl, methoxyphenethyl or hydroxyphenethyl; and R<3> and R<4> are, each, hydroxy, hydrogen, halo, C1-3-alkyl or C1-3alkoxy. The compounds are dopamine agonists and have antihypertensive activity. Pharmaceutical compositions and methods of use are described, as are processes for their preparation.</p>
申请公布号 ES546886(D0) 申请公布日期 1986.10.16
申请号 ES19860005468 申请日期 1985.09.11
申请人 SMITHKLINE BECKMAN CORPORATION 发明人
分类号 A61K31/42;A61K31/423;A61K31/425;A61K31/428;A61P9/08;A61P9/10;A61P9/12;C07D263/58;C07D277/68;(IPC1-7):C07D263/58 主分类号 A61K31/42
代理机构 代理人
主权项
地址