发明名称 2-aminomethyl-6-sulfamoylphenol derivatives, a process for their preparation and their use and also pharmaceutical formulations based on these compounds
摘要 The invention relates to 2-aminomethylphenols of the formula I <IMAGE> in which R1 and R2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl or benzyl which is optionally substituted by alkyl, alkoxy or halogen, R3 and R5 denote hydrogen, halogen, alkyl or alkoxy, R4 denotes halogen, alkyl or cycloalkyl and R6 and R7 represents hydrogen or alkyl, it being possible for the radicals R1 and R2, R6 and R7 and/or two of the radicals R3, R4 and R5 to form an alkylene chain which is optionally substituted by methyl groups and which, in the case of the radicals R1, R2, R6 and R7, can also be interrupted by oxygen atoms, sulfur atoms and/or imino groups, and to physiologically acceptable salts thereof, a process for their preparation, and their use and to pharmaceutical formulations based on these compounds.
申请公布号 US4607030(A) 申请公布日期 1986.08.19
申请号 US19850751995 申请日期 1985.07.03
申请人 HOECHST AKTIENGESELLSCHAFT 发明人 ENGLERT, HEINRICH C.;MANIA, DIETER;MUSCHAWECK, ROMAN;HROPOT, MAX
分类号 A61K31/18;A61K31/40;A61P3/00;A61P7/10;A61P9/12;C07C67/00;C07C301/00;C07C303/02;C07C303/38;C07C303/40;C07C311/15;C07C311/37;C07D295/22;C07D295/26;(IPC1-7):A61K31/40;C07D207/00;C07C143/80 主分类号 A61K31/18
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