发明名称 Aromastase inhibiting alpha , alpha -diarylimidazole-4(5)-propionitriles, alpha , alpha -diarylimidazole-4(5)-propionamides, and 4(5)-(2,2-diarylethyl)imidazoles
摘要 This invention provides a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals by administering certain imidazole derivatives. Pharmaceutical formulations of the imidazole derivatives and certain imidazoles are also provided.
申请公布号 US4605661(A) 申请公布日期 1986.08.12
申请号 US19840621594 申请日期 1984.06.18
申请人 ELI LILLY AND COMPANY 发明人 HIRSCH, KENNETH S.;PIOCH, RICHARD P.
分类号 A61K31/415;A61K31/44;A61K31/4427;A61P35/00;C07D233/54;C07D233/58;C07D233/64;C07D401/06;C12N9/99;(IPC1-7):A61K31/415 主分类号 A61K31/415
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