发明名称 |
Aromastase inhibiting alpha , alpha -diarylimidazole-4(5)-propionitriles, alpha , alpha -diarylimidazole-4(5)-propionamides, and 4(5)-(2,2-diarylethyl)imidazoles |
摘要 |
This invention provides a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals by administering certain imidazole derivatives. Pharmaceutical formulations of the imidazole derivatives and certain imidazoles are also provided.
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申请公布号 |
US4605661(A) |
申请公布日期 |
1986.08.12 |
申请号 |
US19840621594 |
申请日期 |
1984.06.18 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
HIRSCH, KENNETH S.;PIOCH, RICHARD P. |
分类号 |
A61K31/415;A61K31/44;A61K31/4427;A61P35/00;C07D233/54;C07D233/58;C07D233/64;C07D401/06;C12N9/99;(IPC1-7):A61K31/415 |
主分类号 |
A61K31/415 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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