发明名称 PIPERAZINE DERIVATIVE
摘要 NEW MATERIAL:A compound shown by the formula I [R is group shown by the formula II, formula III (R<1> is lower alkoxy, phenyl-substituted lower alkoxy, or phenyl; R<2> is lower alkyl, or phenyl), -S-R<3> (R<3> is phenyl-substituted lower alkyl, phenyl, etc.), or -SO2-R<4> (R<4> is phenyl-substituted lower alkyl or phenacyl)]. EXAMPLE:Diethylpiperazinylamido phosphorate. USE:Useful as a raw material for producing pipemidic acid, norfloxacin, enoxacin, etc., antibacterial agents. PREPARATION:Piperazine is reacted with a compound shown by the formula R-H, to give a compound shown by the formula I.
申请公布号 JPS61176579(A) 申请公布日期 1986.08.08
申请号 JP19850014446 申请日期 1985.01.30
申请人 ROLLER JAPAN KK 发明人 YAHAGI KAZUHIRO;UEMATSU SHIGERU
分类号 C07D295/22;A61K31/495;A61P31/04;C07F9/6509;C07F9/6558;C07F9/6561 主分类号 C07D295/22
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