发明名称 BENZOXAZOLINONES
摘要 <p>The invention relates to compounds of the formula: < IMG > in which R represents hydrogen or a lower alkyl radical and R1 and R2 separately represent hydrogen, a lower alkyl, cycloalkyl or benzyl radical, or represent, together with the nitrogen atom to which they are bonded, a heterocyclic radical such as a morpholino, 4-(pyrimidin-2-yl)-piperazinyl or 4-phenylpiperazinyl the phenyl radical of which being optionally substituted by halogen, lower alkoxy or trifluoromethyl, having CNS activity and particularly hypnotic properties. Moreover the compounds inwhich R1 and R2 are hydrogen can be used in the treatment of heart failure.</p>
申请公布号 CA1208220(A) 申请公布日期 1986.07.22
申请号 CA19830441918 申请日期 1983.11.24
申请人 RIOM LABORATOIRES - CERM S.A. 发明人 CAIGNARD, DANIEL H.;LESPAGNOL, CHARLES;LESIEUR, DANIEL;BUSCH, NORBERT
分类号 A61K31/42;A61K31/423;A61K31/495;A61K31/496;A61K31/505;A61K31/535;A61K31/5377;A61P9/02;A61P9/04;A61P25/00;A61P25/20;C07D263/58;C07D413/12;(IPC1-7):C07D263/58;C07D413/06;C07D413/14 主分类号 A61K31/42
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