发明名称 NEW THIENOPYRIDINE DERIVATIVES,A PROCESS OF PREPARATION THEREOF AND THERAPEUTIC COMPOSITIONS CONTAINING THE SAME
摘要 This invention relates to new derivatives of 5-( omega -phenethylamino-alkyl) -4,5,6,7-tetrahydro-thieno-(3,2-c)-pyridine of the formula <IMAGE> wherein n is an integer of from 2 to 5, R1 represents a hydrogen atom or a 3,4-dimethoxyphenyl group, R2 represents a hydrogen atom, an alkyl group having up to 4 carbon atoms or a 4-cyano-4-(3,4-dimethoxyphenyl)-5-methylhexyl group and R3 represents two or three methoxy groups, to therapeutically acceptable salts thereof, to a process for the preparation of these derivatives comprising condensing a 5-( omega -chloroalkyl)-4,5,6,7- tetrahydro- thieno- (3,2-c)-pyridine with the appropriate phenethyl derivative at from 90 DEG to 130 DEG C. under nitrogen circulation and to therapeutic compositions containing said compounds.
申请公布号 ZA8508267(B) 申请公布日期 1986.06.25
申请号 ZA19850008267 申请日期 1985.10.22
申请人 SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) 发明人 ANDRE ESANU
分类号 A61K31/435;A61P3/00;A61P3/14;A61P7/02;C07D495/04 主分类号 A61K31/435
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