发明名称 FORFARANDE FOR FRAMSTELLNING AV BENSIMIDAZOLDERIVAT
摘要 Benzimidazole derivatives of the formula <IMAGE> in which R and R1 independently of one another are each hydrogen, an alkanoyl group having 1 to 4 carbon atoms, an alkoxycarbonyl group having 1 to 4 carbon atoms, an alkylsulphonyl group having 1 to 4 carbon atoms, a benzoyl group, a phenylsulphonyl group or a p-methylphenylsulphonyl group; R2 and R4 independently of one another are each hydrogen, halogen or a methyl group, R3 is hydrogen, halogen, a methyl group or a methoxy group; X is oxygen or sulphur; Y is halogen, an alkyl group having 1 to 4 carbon atoms, an alkoxy group having 1 to 4 carbon atoms, a methylthio group, a methylsulphinyl group, a methylsulphonyl group, a trifluoromethyl group, a nitro group, a hydroxyl group, a cyano group or an acetyl group; and m is 0, 1, 2 or 3; and if one of the two radicals R or R1 is hydrogen, the position of the other of these radicals on the N atoms cannot be clearly established, including, when at least one of the two radicals R or R1 is hydrogen, the possible tautomeric compounds of the formula I; and the disulphides obtainable by oxidation of compounds of the formula I. The compounds are useful for combating helminths in domestic animals and productive animals.
申请公布号 SE444314(B) 申请公布日期 1986.04.07
申请号 SE19780004058 申请日期 1978.04.11
申请人 CIBA-GEIGY AG 发明人 1)E * AUFDERHAAR;2)J-J * GALLAY;3)M * KUHNE;4)A * MEYER;5)O * RECHSTEINER;6)M * SCHELLENBAUM;7)J-P * FUMEAUX
分类号 A01N43/52;A61K31/415;A61K31/4184;A61P33/00;C07D235/28;(IPC1-7):C07D233/28 主分类号 A01N43/52
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