发明名称 UN PROCEDIMIENTO PARA LA OBTENCION DE PIRIDOINDOLES
摘要 <p>Pyridoindoles of the formula <IMAGE> in which R1 represents hydrogen or C1-C4-alkyl, which is optionally substituted by the radical <IMAGE> R2 and R3 represent H or form a bond, or R1 and R2 together represent O, -O-CH2-CH2-O- or -S-CH2-CH2-S-, R4 represents H or the <IMAGE> or R3 and R4 represent O, or R1 and R4 are members of an N-containing six-membered ring and R8 and R9 represent H or C1-C4-alkyl, or optionally form, with the N atom, a heterocyclic 5-membered or 6-membered ring, which can optionally also contain a further hetero-atom from the series comprising N, O or S, R5 represents H, C1-C4-alkyl or the group <IMAGE> or R5 and R3 form a bond, and R10 and R11 represent C1-C4-alkyl or are members of an N-containing 5-membered or 6-membered ring, R6 represents H or C1-C4-alkyl and R7 represents halogen, or acid addition salts thereof, which are active on the central nervous system. Novel intermediates are also shown.</p>
申请公布号 ES545270(D0) 申请公布日期 1986.03.16
申请号 ES19700005452 申请日期 1985.07.16
申请人 TROPONWERKE GMBH & CO KG 发明人
分类号 A61K31/435;A61K31/445;A61K31/535;A61P25/00;A61P25/20;A61P25/24;A61P25/26;C07C67/00;C07C239/00;C07C251/34;C07D217/04;C07D317/00;C07D471/04;C07D471/14;C07D471/20;C07D491/20;C07D495/20;(IPC1-7):C07D471/04;A61K31/475 主分类号 A61K31/435
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