Disclosed are the compounds of formula (1)in which R1, R7, R8, R9, R10, R17, R18, R19, R20 and m have the meanings as given in the description, which are novel effective inhibitors of type 4 and 5 phosphodiesterase.
申请公布号
EA023713(B1)
申请公布日期
2016.07.29
申请号
EA20140000001
申请日期
2012.06.12
申请人
TAKEDA GMBH
发明人
STENGEL THOMAS;MAIER THOMAS;MANN ALEXANDER;STADLWIESER JOSEF;FLOCKERZI DIETER;PAHL ANDREAS;BENEDIKTUS EWALD;HESSMANN MANUELA;KANACHER TOBIAS;HUSSONG RAGNA;ZITT CHRISTOF;HOLST HANS, CHRISTOF;HUMMEL ROLF-PETER;VIERTELHAUS MARTIN;TENOR HERMANN;DUNKERN TORSTEN;HATZELMANN ARMIN;HESSLINGER CHRISTIAN