发明名称 PROCESS FOR THE PREPARATION OF BETA-CYCLO-SUBSTITUTED ETHYL AMINES, AND PRODUCTS SO OBTAINED
摘要 The present invention provides a multistep process for the preparation of beta -cyclo-substituted ethylamines of the general formula:- Ar-CH2-CH2-NH2 +TM, (I) in which AR is a heterocyclic or non-heterocyclic aromatic radical, which is optionally mono- or poly- substituted, wherein said compounds represent a class of intermediates which can be converted to 4,5,6,7-tetrahydro[3,2-C] or [2,3-C]pyridines wherein the latter are useful for anti-inflammatory, vasodilator or blood platelet aggregation inhibition activities.
申请公布号 DE3266363(D1) 申请公布日期 1985.10.24
申请号 DE19823266363 申请日期 1982.06.18
申请人 SANOFI, SOCIETE ANONYME 发明人 CHEKROUN, ISAAC;HEYMES, ALAIN
分类号 C07C67/00;C07C209/00;C07C209/62;C07C209/68;C07C211/27;C07C213/00;C07C217/60;C07D213/38;C07D307/52;C07D307/54;C07D333/20;C07D333/28;C07F9/24;C07F9/40;C07F9/58;C07F9/655;C07F9/6553;(IPC1-7):C07C85/24;C07C87/28;C07D213/18 主分类号 C07C67/00
代理机构 代理人
主权项
地址