发明名称 N-((2-AMINO-5-HALO-6-(SUBSTITUTED)-3-PYRAZINYL)-METHYLENE)AMINE ANTIMICROBIAL COMPOUNDS
摘要 Antimicrobial compounds of the formula: <IMAGE> (I.) wherein: Hal is bromine or chlorine; R is halo; mono- or di-substituted mono- or diloweralkylamino wherein the loweralkyl substituents are hydroxy or loweralkanoyloxy; 4-morpholino; thiocyano; mercapto; straight or branched chain C1-8alkylthio; mono- or di-substituted loweralkylthio wherein the substituents are hydroxy, amino, loweralkanoylamino, or loweralkoxycarbonyl; arylthio; loweralkylsulfoxy; or loweralkylsulfonyl; R1 is hydrogen; straight or branched C1-8alkyl; aryl; aryl substituted with up to two members selected from the group consisting of C1-3alkyl, C1-3alkoxy, halo, and mono- or di-C1-3alkyl substituted amino; heteroaryl; formyl C2-4alkenyl; or C2-4alkenyl; and R2 is straight or branched C1-8alkyl; loweralkoxy; hydroxy; loweralkoxycarbonylmethyl; benzyl; or benzyl substituted with up to two members selected from the group consisting of halo, loweralkyl, and loweralkoxy; are useful in various agricultural and industrial areas.
申请公布号 ZA8309540(B) 申请公布日期 1985.08.28
申请号 ZA19830009540 申请日期 1983.12.22
申请人 MERCK & CO.,INC. 发明人 DAVID B.R. JOHNSTON
分类号 A01N43/60;C07D241/20 主分类号 A01N43/60
代理机构 代理人
主权项
地址