发明名称 3-SUBSTITUTED-2-OXO-1-AZETIDINE SULPHONIC ACID DERIVATIVES
摘要 <p>Beta lactams (I) having an SO3M substit. at 1-position and an opt. substd. or protected amino gp. or azido gp. at the 3-position are new. (M is hydrogen or a cation). They can also be substd. at the 4-position by alkyl, cycloalkyl, opt. substd. phenyl, alkoxycarbonyl, alken-1-yl, alkyn-1-yl, 2-phenylethenyl or 2-phenylethynyl. (I) having a 3-acylamino substit. are antibacterials effective against Gram negative and positive species, and useful therapeutically in human or veterinary medicine. The other new cpds. are intermediates.</p>
申请公布号 HK57785(A) 申请公布日期 1985.08.09
申请号 HK19850000577 申请日期 1985.08.01
申请人 E. R. SQUIBB & SONS INC. 发明人 RICHARD BROOK SYKES;WILLIAM LAWRENCE PARKER;CHRISTOPHER MICHAEL CIMARUSTI;WILLIAM HENRY KOSTER;WILLIAM ALLEN SLUSARCHYK;ALAN WILLIAM FRITZ;DAVID MACK FLOYD
分类号 A61K31/395;A61K31/397;A61K31/41;A61K31/42;A61K31/425;A61K31/435;A61P31/04;C07C67/00;C07C301/00;C07C303/34;C07C307/02;C07D205/08;C07D205/085;C07D213/18;C07D401/12;C07D401/14;C07D403/12;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D417/12;C07D471/04;C07F7/08;C07F7/10;C07F9/6558;C12P17/10;(IPC1-7):C07D205/08;C07D401/00;C07D403/02;C07D405/00;C07D409/00;C07D413/02;C07D417/00;C07D471/00 主分类号 A61K31/395
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