发明名称 Phosphorinane deriv.
摘要 <p>3-(2-Chloroethyl) 2-((2-chloroethyl)amino) 1,3,2-oxaza phosphorinano-2-oxide of formula (I) is made by (a) reacting a cpd. of formula (II) with 3-halo propanol to obtain a cpd. of formula (III); (b) this is reacted with phosphorus oxychloride to obtain 2-chloro 3-(2-chloroethyl) 1,3,2-oxazaphosphorinano-2-oxide; and (c) this cpd. is reacted with 2-chloroethylamine hydrochloride to give (I).</p>
申请公布号 ES8504835(A3) 申请公布日期 1985.07.16
申请号 ES19940005261 申请日期 1983.10.03
申请人 SOC. ESP. ESPECIALIDADES FARMACO-TERAPEUTICAS S.A. 发明人
分类号 (IPC1-7):C07F9/65 主分类号 (IPC1-7):C07F9/65
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