发明名称 20-AMINO MACROLIDE DERIVATIVES
摘要 Compds. of formula (I) and their acid addn. salts are new. In the formula (I), R is a mono-, bi-, or tricyclic opt. unsatd. ring contg. 1N as sole heteroatom and bonded through the N; R1 is H or an OH protecting gp.; R2 is H, C1-5 alkanoyl, PhCH2W, PhC2H4CO, or PhCO2; R3 is H, iodo, OH, mycarosyloxy, or C1-5 alkanoyloxy; and R4 is mycinoxyloxy. Compds. (I) are broad-spectrum antibacterials and are effective against Pasteurella and Mycoplasma species, e.g. causing mycoplasmal pneumonia in swine.
申请公布号 KR850000961(B1) 申请公布日期 1985.07.02
申请号 KR19830004273 申请日期 1983.09.12
申请人 ELI LILLY AND CO. 发明人 DEBONO, MANUEL;KIRST, HERBERT ANDREW
分类号 C07D313/00;A23K20/195;A61K31/70;A61K31/7042;A61K31/7048;A61P31/04;C07D309/36;C07D315/00;C07H15/00;C07H17/08 主分类号 C07D313/00
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