发明名称 N-Pyrazolylalkylenediamine intermediates
摘要 New N-heteroarylalkylenediamine <IMAGE> wherein R1 and R2 each independently is hydrogen, an alkyl radical containing up to 6 carbon atoms, or a benzyl radical, X is an alkylene radical containing 2 to 6 carbon atoms, A is a mono- or bicyclic heteroaromatic radical, which can be partly hydrogenated, with the proviso that it contains 2 or 3 adjacent ring heteroatoms, whereby the bound ring heteroatoms can be an oxygen atom and a nitrogen atom or 2 or 3 nitrogen atoms, and R3, R4, R5, R6 and R7 each independently is hydrogen, or an alkyl radical containing up to 6 carbon atoms, which can be substituted by hydroxyl, carbamyl, nitrile or carboxyl, an alkenyl radical containing 2 to 6 carbon atoms, a phenyl or carbamyl radical or one of the divalent substituents oxygen or sulphur, or a salt thereof. The compounds are intermediates in the synthesis of cardioactive compounds.
申请公布号 US4507488(A) 申请公布日期 1985.03.26
申请号 US19830483788 申请日期 1983.04.11
申请人 BOEHRINGER MANNHEIM GMBH 发明人 WIEDEMANN, FRITZ;RIEGER, EWALD
分类号 A61K31/38;A61K31/045;A61K31/135;A61K31/138;A61K31/40;A61K31/41;A61K31/415;A61K31/435;A61K31/47;A61K31/472;A61K31/473;A61K31/495;A61K31/498;A61K31/50;A61K31/505;A61K31/52;A61K31/522;A61P9/00;A61P9/04;C07C217/32;C07C217/72;C07C217/78;C07C219/06;C07C219/08;C07C219/14;C07D209/48;C07D213/74;C07D215/46;C07D217/22;C07D219/12;C07D231/06;C07D231/20;C07D231/32;C07D231/38;C07D231/46;C07D231/52;C07D231/56;C07D237/20;C07D239/42;C07D239/54;C07D239/545;C07D239/557;C07D239/56;C07D239/84;C07D239/95;C07D241/44;C07D249/18;C07D333/36;C07D473/16;C07D473/32;C07D473/34;C07D487/00;C07D487/04;(IPC1-7):C07D231/38 主分类号 A61K31/38
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