摘要 |
<p>A compound of the formula:
<Chemistry id="chema01" num="0001"><Image id="ia01" he="35" wi="39" file="IMGA0001.TIF" imgContent="chem" imgFormat="TIFF" inline="no" /></Chemistry>(wherein Az is imidazolyl or triazolyl;
<UnorderedLists id="ula01" listStyle="none"><ListItem>R is C<Sub>1</Sub>-C<Sub>5</Sub> Alkyl or phenyl optionally substituted by 1 to 3 members selected from halogen, C<Sub>1</Sub>-C<Sub>5</Sub> alkyl, and C<Sub>1</Sub>-C<Sub>5</Sub> alkoxy;</ListItem><ListItem>X<Sup>1</Sup> and X<Sup>2</Sup> each is hydrogen, halogen, C<Sub>1</Sub>-C<Sub>5 </Sub>alkyl, or C<Sub>1</Sub>-C<Sub>5</Sub> alkoxy;</ListItem><ListItem>Y is C=O, C = S, S=O, or R<Sup>1</Sup>-C-R<Sup>2</Sup>; and</ListItem><ListItem>R' and R<Sup>2</Sup> each is hydrogen, C,-C<Sub>3</Sub> alkyl or, taken together may form C<Sub>4</Sub>-C<Sub>6</Sub> alkylene) or its acid addition salt being useful as an antimycotic agent is prepared by reacting a corresponding diol with a cyclizing agent.</ListItem></UnorderedLists></p> |