发明名称 |
Beta-lactamase inhibiting 6-(alkoxyamino-methyl) penicillanic acid 1,1-dioxide and derivatives |
摘要 |
6-alpha/beta-[(C1-C4)Alkoxyaminomethyl and benzyloxyaminomethyl]penicillanic acid 1,1-dioxides, pharmaceutically acceptable salts thereof and conventional esters thereof hydrolyzable under physiological conditions, all of which are useful in medicine as beta-lactamase inhibitors; intermediates and processes therefor; and a process for the conversion of the present compounds to 6-alpha- and 6-beta-(aminomethyl)penicillanic acid 1,1-dioxides and derivatives.
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申请公布号 |
US4499017(A) |
申请公布日期 |
1985.02.12 |
申请号 |
US19830501475 |
申请日期 |
1983.06.06 |
申请人 |
PFIZER INC. |
发明人 |
PIRIE, DONALD K.;VOLKMANN, ROBERT A.;KLEINMAN, EDWARD F. |
分类号 |
C07D499/87;A61K31/43;A61P31/04;C07D499/00;C07D499/86;C07D499/861;C07D499/897;(IPC1-7):C07D499/00;A61K31/415 |
主分类号 |
C07D499/87 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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