发明名称 |
PROCESS FOR PREPARING PYRIMIDINE DERIVATIVES |
摘要 |
The pyrimidine derivatives of formula I <IMAGE> I wherein R1 is naphthyl, substituted naphthyl or substituted phenyl; R2 is hydrogen or lower alkoxy; and A is an optionally present ethylene or 1,3-propylene, and wherein the diaminopyridine group has the exo-configuration when A is present, are described. These compounds are useful as antibacterial agents, antimalarial agents and antitumor agents, and can be used in combination with sulfonamides in the control of bacterial infections. |
申请公布号 |
HUT34017(A) |
申请公布日期 |
1985.01.28 |
申请号 |
HU19840001409 |
申请日期 |
1984.04.11 |
申请人 |
F.HOFFMANN-LA ROCHE ET CO,AG,CH |
发明人 |
KOMPIS,IVAN,CH;LOCHER,RITA,CH;MAAG,HANS,CH |
分类号 |
A61K31/505;C07D211/70;C07D211/74;C07D211/78;C07D401/04;C07D451/02;C07D451/06;C07D451/14 |
主分类号 |
A61K31/505 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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