发明名称 WERKWIJZE VOOR HET BEREIDEN VAN ANTI-TUMOR-MIDDELEN EN DAARVOOR GESCHIKTE GENEESKRACHTIGE VERBINDINGEN.
摘要 The known antitumor antibiotic adriamycin and its beta -anomer, and the novel compounds, 4'-epiadriamycin (both alpha - and beta -anomers) are prepared by condensing a novel, reactive protected derivative of adriamycinone with reactive intermediates which are 1-halo-2,3,6-trideoxy-3-trifluoroacetamido-4-trifluoroacetoxy- alpha -L-lyxo (or arabino) hexopyranoses.
申请公布号 NL176635(B) 申请公布日期 1984.12.17
申请号 NL19750002934 申请日期 1975.03.12
申请人 FARMITALIA CARLO ERBA S.P.A. TE MILAAN, ITALIE. 发明人
分类号 C07H15/24;A61K31/70;A61K31/7028;A61K31/7034;A61K31/704;A61P35/00;C07H15/252;(IPC1-7):61K31/70;07H15/24 主分类号 C07H15/24
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