发明名称 |
Iodinated vasopressin antagonists |
摘要 |
A series of vasopressin antagonists which have a 3'-iodo-tyrosine unit at position 2 are prepared by iodination of the tyrosine congeners. The compounds have antagonist activity manifested by an aquaretic effect and, also, are useful in studying various biological reactions.
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申请公布号 |
US4469680(A) |
申请公布日期 |
1984.09.04 |
申请号 |
US19830511120 |
申请日期 |
1983.07.06 |
申请人 |
SMITHKLINE BECKMAN CORPORATION |
发明人 |
HUFFMAN, WILLIAM F.;MOORE, MICHAEL L. |
分类号 |
A61K38/00;C07K7/16;(IPC1-7):A61K37/00;A61K43/00;G01N33/00;C07C103/52 |
主分类号 |
A61K38/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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