发明名称 |
INTERMEDIATES FOR THE PREPARATION OF THIENAMYCIN AND PROCESS FOR PREPARING INTERMEDIATES |
摘要 |
<p>In a process for the total synthesis of thienamycin from L-aspartic acid via intermediate III: <CHEM> R = H, blocking group or salt cation there is disclosed a process for preparing III via <CHEM> wherein R is a protecting group.</p> |
申请公布号 |
EP0026816(B1) |
申请公布日期 |
1984.05.30 |
申请号 |
EP19800104296 |
申请日期 |
1980.07.22 |
申请人 |
MERCK & CO. INC. |
发明人 |
CHRISTENSEN, BURTON G.;RATCLIFFE, RONALD W.;SALZMANN, THOMAS N. |
分类号 |
C07D499/06;A61K31/395;A61K31/397;A61P31/04;C07D205/08;C07D477/00;C07D477/04;C07D477/10;C07F7/10;(IPC1-7):07D205/08;07F7/10 |
主分类号 |
C07D499/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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