发明名称 CYSTEIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM
摘要 1. Cysteine derivatives having the general formula see diagramm : EP0035641,P15,F1 wherein R represents hydrogen, an alkyl radical having from 1 to 4 carbon atom(s), an alkali or alkaline-earth metal or a quaternary ammonium group, R1 means an alkyl carbonyl radical having from 2 to 4 carbon atoms, a 2-(6'-methoxynapht-2'-yl)-propionyl radical or a 2-(2'-ethyl-2',3'-dihydro benzofuran-5'-yl)- acetyl radical and R2 represents hydrogen, a 2-(6'-methoxynapht-2'-yl)- propionyl radical or a 2-(2'-ethyl-2',3'-dihydrobenzofuran- 5'-yl)-acetyl radical, with the further definitions that a) in case that one of R1 and R2 represents a 2-(6'-methoxynapht-2'-yl)- propionyl radical or a 2-(2'-ethyl-2',3'-dihydrobenzofuran- 5'-yl)-acetyl radical, the other one of R1 and R2 is different from a 2-(6'-methoxynapht-2'-yl)-propionyl radical and 2-(2'-ethyl-2',3'-dihydrobenzofuran-5'-yl)-acetyl radical and b) in case that R1 represents an alkyl carbonyl radical having from 2 to 4 carbon atoms R2 is different form hydrogen in the form of the separated optically active isomers or of mixtures of them.
申请公布号 DE3163254(D1) 申请公布日期 1984.05.30
申请号 DE19813163254 申请日期 1981.01.30
申请人 ALFA FARMACEUTICI S.P.A. 发明人 MASCELLANI, GIUSEPPE;TAMAGNONE, GIANFRANCO;GUERRA, GUIDO;BENELLI, AUGUSTA
分类号 A61K31/195;A61K31/198;A61K31/22;A61K31/34;A61K31/343;A61P25/04;A61P29/00;C07C67/00;C07C313/00;C07C323/59;C07C325/00;C07C327/20;C07D307/79;C07F7/18;(IPC1-7):C07C149/24;A61K31/19 主分类号 A61K31/195
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