| 摘要 |
<p>…<CHEM>… Piperidyl N-(4-quinolyl)-anthraniloyloxyalkanoates I and their pharmaceutically acceptable salts in which… R = C1-C4 alkyl, (straight or branched), C2C6 alkenyl, C2C6 alkynyl, benzyl, phenethyl, 4-nitro-phenethyl or 4-amino-phenethyl; or phenacyl, benzoylethyl, beta -hydroxyphenethyl or alpha -hydroxy-phenylpropyl, optionally substituted in the phenyl ring by one or more of a halogen atom, CF3, NO2, NH2, C1-C4 alkyl or C1-C4 alkoxy,… R1 = H or phenyl… R2 = H or C1-C4 alkyl… R3 = H or C1-C4 alkyl… one of R4 and R5 = Cl or CF3 and… the other of R4 and R5 = H… have analgesic and antiinflammatory properites. They are also inhibitors of platelet aggregation and anti-depressant agents. Their preparation and pharmaceutical compositions containing them are also disclosed.</p> |
