发明名称 [2-(5-Nitro-2-furyl)-vinyl]-pyrimidin-Derivate und Verfahren zu deren Herstellung
摘要 <FORM:1113382/C2/1> Novel compounds of Formula I, in which R is a C1- 4 alkylthio, amino, C1- 4 alkylamino, di-(C1- 4 alkyl) amino or C1- 4 alkanoylamino group and R1 is a hydrogen atom or a C1- 4 alkyl group are prepared by condensing 5-nitrofurfural, or its diacetate, with a compound of the Formula II, preferably in the presence of a dehydrating agent. When an anhydride of a carboxylic acid of 1-4 carbon atoms is used as the dehydrating agent, compounds in which R is a C1- 4 alkanoyl-amino group are obtained from starting materials in which R is NH2. The compounds in which R is an alkanoylamino group are also obtained by acylating the corresponding amino compounds. The compounds in which R is an amino group may be obtained by hydrolysis of the corresponding acylamino compounds.
申请公布号 DE1670532(A1) 申请公布日期 1970.11.12
申请号 DE19661670532 申请日期 1966.08.31
申请人 DAINIPPON PHARMACEUTICAL COMPANY LTD. 发明人 MINAMI,SHINSAKU;FUJITA,AKIE;SHIMIZU,MASANAO;TAKASE,YOSHIYUKI
分类号 C07D405/06;C09B51/00 主分类号 C07D405/06
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